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Enzymatic Synthesis of New Acetoacetate–Ursodeoxycholic Acid Hybrids as Potential Therapeutic Agents and Useful Synthetic Scaffolds as Well
Venturi, Valentina; Marchesi, Elena; Perrone, Daniela; Costa, Valentina; Catani, Martina; Aprile, Simona; Lerin, Lindomar Alberto; Zappaterra, Federico; Giovannini, Pier Paolo; Preti, Lorenzo     dettagli >>
MOLECULES
Vol. 29, No. 6, pp: 1305-1314, Anno: 2024

Dihydroartemisinin-Ursodeoxycholic Bile Acid Hybrids in the Fight against SARS-CoV-2
Marchesi, E.; Gentili, V.; Bortolotti, D.; Preti, L.; Marchetti, P.; Cristofori, V.; Fantinati, A.; Rizzo, R.; Trapella, C.; Perrone, D.; Navacchia, M. L.     dettagli >>
ACS OMEGA
Vol. 8, No. 47, pp: 45078-45087, Anno: 2023

Molecular Hybridization as a Strategy for Developing Artemisinin-Derived Anticancer Candidates
Marchesi, Elena; Perrone, Daniela; Navacchia, Maria Luisa     dettagli >>
PHARMACEUTICS
Vol. 15, No. 9, pp: 2185-2226, Anno: 2023

Anticancer Activity and Molecular Mechanisms of an Ursodeoxycholic Acid Methyl Ester-Dihydroartemisinin Hybrid via a Triazole Linkage in Hepatocellular Carcinoma Cells
Hsu, Ya-Fen; Kung, Fan-Lu; Huang, Tzu-En; Deng, Yi-Ning; Guh, Jih-Hwa; Marchetti, Paolo; Marchesi, Elena; Perrone, Daniela; Navacchia, Maria Luisa; Hsu, Lih-Ching     dettagli >>
MOLECULES
Vol. 28, No. 5, pp: 2358-2374, Anno: 2023

Synthesis and Biological Investigation of Bile Acid-Paclitaxel Hybrids
Melloni, E.; Marchesi, E.; Preti, L.; Casciano, F.; Rimondi, E.; Romani, A.; Secchiero, P.; Navacchia, M. L.; Perrone, D.     dettagli >>
MOLECULES
Vol. 27, No. 2, pp: 471-1-471-15, Anno: 2022

Organocatalytic synthesis of poly(hydroxymethylfuroate) via ring-opening polymerization of 5-hydroxymethylfurfural-based cyclic oligoesters
Ragno, Daniele; Di Carmine, Graziano; Vannini, Micaela; Bortolini, Olga; Perrone, Daniela; Buoso, Sara; Bertoldo, Monica; Massi, Alessandro     dettagli >>
POLYMER CHEMISTRY
Vol. 13, No. 10, pp: 1350-1358, Anno: 2022

Antisense oligonucleotides conjugated with lipophilic compounds: synthesis and in vitro evaluation of exon skipping in duchenne muscular dystrophy
Marchesi, E.; Cortesi, R.; Preti, L.; Rimessi, P.; Sguizzato, M.; Bovolenta, M.; Perrone, D.     dettagli >>
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
Vol. 23, No. 8, pp: 4270-1-4270-21, Anno: 2022

Synthesis of 2,6-Dimethyltyrosine-Like Amino Acids through Pinacolinamide-Enabled C-H Dimethylation of 4-Dibenzylamino Phenylalanine
Illuminati, D.; Fantinati, A.; De Ventura, T.; Perrone, D.; Sturaro, C.; Albanese, V.; Marzola, E.; Cristofori, V.; Oble, J.; Poli, G.; Trapella, C.     dettagli >>
JOURNAL OF ORGANIC CHEMISTRY
Vol. 87, No. 5, pp: 2580-2589, Anno: 2022

Synthesis and exon‐skipping properties of a 3′‐ursodeoxycholic acid‐conjugated oligonucleotide targeting dmd pre‐mrna: Pre‐synthetic versus post‐ synthetic approach
Marchesi, E.; Bovolenta, M.; Preti, L.; Capobianco, M. L.; Mamchaoui, K.; Bertoldo, M.; Perrone, D.     dettagli >>
MOLECULES
Vol. 26, No. 24, pp: 7662-7678, Anno: 2021

Bile Acid Conjugates with Anticancer Activity: Most Recent Research
Navacchia, Maria Luisa; Marchesi, Elena; Perrone, Daniela     dettagli >>
MOLECULES
Vol. 26, No. 1, pp: 25-1-25-19, Anno: 2021

Modified nucleosides, nucleotides and nucleic acids via click azide-alkyne cycloaddition for pharmacological applications
Perrone, D.; Marchesi, E.; Preti, L.; Navacchia, M. L.     dettagli >>
MOLECULES
Vol. 26, No. 11, pp: 3100-1-3100-27, Anno: 2021

Evaluation of the Anticancer Activity of a Bile Acid-Dihydroartemisinin Hybrid Ursodeoxycholic-Dihydroartemisinin in Hepatocellular Carcinoma Cells
Huang, T. -E.; Deng, Y. -N.; Hsu, J. -L.; Leu, W. -J.; Marchesi, E.; Capobianco, M. L.; Marchetti, P.; Navacchia, M. L.; Guh, J. -H.; Perrone, D.; Hsu, L. -C.     dettagli >>
FRONTIERS IN PHARMACOLOGY
Vol. 11, No. 1, pp: 599067-1-599067-14, Anno: 2020

Oligonucleotides: Current Trends and Innovative Applications in the Synthesis, Characterization, and Purification
Catani, Martina; DE LUCA, Chiara; Medeiros Garcia Alcântara, Joao; Manfredini, Nicolò; Perrone, Daniela; Marchesi, Elena; Weldon, Richard; Müller-Späth, Thomas; Cavazzini, Alberto; Morbidelli, Massimo; Sponchioni, Mattia     dettagli >>
BIOTECHNOLOGY JOURNAL
Vol. 15, No. 8, pp: 1900226-1-1900226-14, Anno: 2020

LSD1 is an environmental stress-sensitive negative modulator of the glutamatergic synapse
Longaretti, A.; Forastieri, C.; Toffolo, E.; Caffino, L.; Locarno, A.; Miseviciute, I.; Marchesi, E.; Battistin, M.; Ponzoni, L.; Madaschi, L.; Cambria, C.; Bonasoni, M. P.; Sala, M.; Perrone, D.; Fumagalli, F.; Bassani, S.; Antonucci, F.; Tonini, R.; Francolini, M.; Battaglioli, E.; Rusconi, F.     dettagli >>
NEUROBIOLOGY OF STRESS
Vol. 13, No. 1, pp: 100280-1-100280-13, Anno: 2020

Dihydroartemisinin-Bile Acid Hybridization as an Effective Approach to Enhance Dihydroartemisinin Anticancer Activity
Marchesi, E.; Chinaglia, N.; Capobianco, M. L.; Marchetti, P.; Huang, T. -E.; Weng, H. -C.; Guh, J. -H.; Hsu, L. -C.; Perrone, D.; Navacchia, M. L.     dettagli >>
CHEMMEDCHEM
Vol. 14, No. 7, pp: 779-787, Anno: 2019

A New Drug Delivery System Based on Tauroursodeoxycholic Acid and PEDOT
Carli, S; Fioravanti, Giulia; Armirotti, A; Ciarpella, F; Prato, M; Ottonello, G; Salerno, M; Scarpellini, A; Perrone, D; Marchesi, E; Ricci, D; Fadiga, L     dettagli >>
Wiley-VCH Verlag, CHEMISTRY-A EUROPEAN JOURNAL
Vol. 25, No. 9, pp: 2322-2329, Anno: 2019

UDP-GlcNAc Analogues as Inhibitors of O-GlcNAc Transferase (OGT): Spectroscopic, Computational, and Biological Studies
Ghirardello, Mattia; Perrone, Daniela; Chinaglia, Nicola; Sádaba, David; Delso, Ignacio; Tejero, Tomas; Marchesi, Elena; Fogagnolo, Marco; Rafie, Karim; van Aalten, Daan M. F.; MERINO FILELLA, PEDRO JOSE     dettagli >>
CHEMISTRY-A EUROPEAN JOURNAL
Vol. 24, No. 28, pp: 7264-7272, Anno: 2018

Conjugated Oligonucleotides for Biochemical Applications
L Capobianco, Massimo; Luisa Navacchia, Maria; Marchesi, Elena; Perrone, Daniela     dettagli >>
MEDICINAL CHEMISTRY
Vol. 7, No. 7, pp: 933-943, Anno: 2017

Fluorous-tag assisted synthesis of bile acid-bisphosphonate conjugates via orthogonal click reactions: an access to potential anti-resorption bone drugs
Massarenti, C.; Bortolini, O.; Fantin, G.; Cristofaro, D.; Ragno, D.; Perrone, D.; Marchesi, E.; Toniolo, Giandomenico; Massi, A.     dettagli >>
ORGANIC & BIOMOLECULAR CHEMISTRY
Vol. 15, No. 22, pp: 4907-4920, Anno: 2017

Exploring Splicing-Switching Molecules For Seckel Syndrome Therapy
Scalet, Daniela; Balestra, Dario; Rohban, Sara; Bovolenta, Matteo; Perrone, Daniela; Bernardi, Francesco; Campaner, Stefano; Pinotti, Mirko     dettagli >>
BIOCHIMICA ET BIOPHYSICA ACTA. MOLECULAR BASIS OF DISEASE
Vol. 1863, No. 1, pp: 15-20, Anno: 2017

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